Nonsteroidal progesterone receptor ligands. 1. 3-Aryl-1-benzoyl-1,4,5,6-tetrahydropyridazines

J Med Chem. 1995 Dec 8;38(25):4878-9. doi: 10.1021/jm00025a003.
No abstract available

MeSH terms

  • Animals
  • Drug Design
  • Female
  • Ligands
  • Progestins / metabolism
  • Promegestone / metabolism
  • Pyridazines / chemical synthesis
  • Pyridazines / metabolism*
  • Pyridazines / pharmacology
  • Rabbits
  • Receptors, Progesterone / metabolism*
  • Structure-Activity Relationship
  • Uterus / metabolism

Substances

  • Ligands
  • Progestins
  • Pyridazines
  • Receptors, Progesterone
  • Promegestone